Kiwon lafiyaShirye-shirye

"Oseltamivir": umarnin don amfani, analogs, bayanin da miyagun ƙwayoyi

Me rubũta da miyagun ƙwayoyi "Oseltamivir"? Umarnin don amfani, analogs, alamomi da contraindications da miyagun ƙwayoyi za a iya bayyana kadan kara. Mu kuma gaya muku game da tsari a cikin abin da za ka iya saya ce medicament, abin da kaddarorin shi yana da, ko illa da sauransu. D.

A siffar, tsari da bayanin da miyagun ƙwayoyi

A sayar da miyagun ƙwayoyi zo a cikin nau'i na rawaya-fari capsules. "Oseltamivir" - shi ne mai prodrug. Lokacin da ingested, shi ne hydrolyzed da kuma tuba zuwa ga aiki sashi - oseltamivir carboxylate.

Bugu da kari ga capsules da medicament aka sallami a cikin nau'i na wani haske foda na baka dakatar.

Features magani

miyagun ƙwayoyi "Oseltamivir" Yaya ta yi aiki? Umarnin a kan aikace-aikace ya furta cewa, da warkewa sakamako na wannan magani dogara ne a kan danniya na aiki na enzymes, wanda aka located a farfajiya na virion mura cutar.

A kan samu na medicament a cikin jikin mutum ta kuriyar ne sāke zuwa aiki metabolite. Saboda haka, oseltamivir carboxylate selectively damuarn neuraminidase. A sakamakon irin wannan daukan hotuna ceases kwayar cell multiplication tsari.

Bisa ga art, shan wannan magani ya kamata a gudanar a cikin 35 hours bayan na farko da ãyõyin mura. Kawai a cikin wannan hanya da tsawon da cutar za a iya rage da kashi 30%, da kuma yiwuwar samun rikitarwa da kuma tsananin cututtuka - 40%.

Pharmacokinetics da miyagun ƙwayoyi

Ko magani ne tunawa "Oseltamivir"? Umurnai na amfani nuna cewa game da 90% na oseltamivir phosphate tunawa a cikin gastro-na hanji fili. The aiki abu ne tuba zuwa carboxylate na oseltamivir, sa'an nan ya shiga cikin tsari dabam dabam.

Game da 3% na aiki sashi yana daure wa jini sunadaran. Its bioavailability ne kamar 76-85% da kuma kawar rabin-rai - 120 minti.

Daga adam oseltamivir carboxylate aka samu ta hanyar da kodan (kamar 80%) kuma Gut (20%). Half-rai da miyagun ƙwayoyi ne 6-10 hours.

alamomi

Me rubũta da miyagun ƙwayoyi "Oseltamivir" (farm kungiyar -. Antiviral jamiái)? Bisa ga umarnin, da medicament da ake amfani da su bi da mura A da B. Har ila yau, shi ne sau da yawa amfani rigakafin kwayar cututtuka.

contraindications

Shin Contra "Oseltamivir" (bayanin irin shirye-shiryen da aka gabatar a sama)? Bisa ga umarnin, da miyagun ƙwayoyi shan da aka haramta a:

  • Hypersensitivity zuwa aiki sashi.
  • koda gazawar (aminci da kuma inganci na da miyagun ƙwayoyi a wadannan marasa lafiya ba a gano).
  • a cikin yara, matasa, fiye da shekara 1 (akwai rashin tabbas kamar yadda ga samuwar na BBB a yara).
  • ciki da kuma nono (shi ba a san ko da miyagun ƙwayoyi ne excreted a nono na mata, da kuma ko yana rinjayar da tayin).

Ya kamata kuma a lura cewa wannan magani ba da shawarar yara a karkashin shekaru 13, kamar yadda masana sun ba aka ƙaddara lafiya da kuma inganci na 'Oseltamivir' domin yin rigakafi da magani na mura.

Drug "Oseltamivir": umarnin don amfani da

Vidal (Magunguna Handbook) ya ƙunshi cikakken bayani a kan yadda kuma a cikin abin da sashi ya kamata ka dauki da miyagun ƙwayoyi a tambaya. Duk da haka, ya kamata a lura da cewa rubũta da miyagun ƙwayoyi ya kamata kawai likita. Bayan duk, kawai wani gogaggen gwani zai iya zabi da hakkin magani regimen, abin da sauri kuma yadda ya kamata kashe duk m bayyanar cututtuka na kwayar cutar.

Saboda haka a cikin abin da sashi An wajabta "Oseltamivir"? Umarnin don amfani a nuna cewa wannan magani ya kamata a yi amfani a cikin kwanaki 2 bayan da farko na farko alamun da mura.

Yara girmi shekaru 13 da kuma manya da miyagun ƙwayoyi gudanar a wani adadin na 75 MG sau biyu a rana kwanaki 5. Ya kamata a lura da cewa, nan da nan kara da sashi daga cikin miyagun ƙwayoyi (msl, har zuwa 150 MG da rana) bai kai ga ya karu warkewa sakamako.

Idan da miyagun ƙwayoyi kana so ka sanya ga yara shekaru 1-12 shekaru, da sashi ne gyara dangane da yaro ta jiki nauyi.

Don hana mura zuwa manya da yara sama da shekaru 13 wajabta 75 MG 1 zarar for 6 makonni a cikin yini (misali, a lokacin da annoba).

Marasa lafiya da CL creatinine kasa da 30 ml da minti bukata gyara sashi (75 MG da zarar kwanaki 5 a kowace rana).

Side effects da miyagun ƙwayoyi bayan ingestion

Duk wani m halayen faruwa bayan gwamnatin 'Oseltamivir' shiri? Umarnin a kan aikace-aikace ce da aka fi bayyana m halayen ne tashin zuciya da kuma amai. A mafi yawan lokuta, wadannan effects ne m, ko moderately bayyana kuma yawanci faruwa a farkon kwanaki da magani.

Ya kamata kuma a lura da cewa a wasu marasa lafiya, a marasa lafiya karbar magani a karkashin review, ci gaba mashako, vertigo, rashin barci, m angina, pseudomembranous colitis, anemia, ciwon huhu, karayar humerus, peritonsillar ƙurji da kuma zazzabi.

Very rare a mutanen da shan miyagun ƙwayoyi "Oseltamivir", akwai ciwon mara, ciwon ji, nosebleeds da conjunctivitis. A mafi yawan lokuta, wadannan halayen faruwa ne kawai sau daya da kuma bace a kan nasu, duk da ci gaba da far. Irin mamaki ba ya bukatar an daina shan magani.

Wadannan da nada antiviral miyagun ƙwayoyi a yara da kuma matasa ma bayyananniya illa. Wadannan sun hada da irin abubuwan da kurji, mai guba epidermal necrolysis, kumburi na harshe, ko fuska, arrhythmia, da ruɗewa, seizures da kuma worsening da ciwon sukari kwarara.

miyagun ƙwayoyi interactions

Bayani samu a cikin shakka daga cikin pharmacokinetic kuma pharmacological nazarin bayyana cewa ci gaban da asibiti gagarumin miyagun ƙwayoyi interactions da wannan miyagun ƙwayoyi ne mai wuya.

The umarnin hada da miyagun kwayoyi, aka ce cewa lokaci daya aikace-aikace na medicament da probenecid take kaiwa zuwa wani karuwa a AUC na aiki metabolite na 2 sau. Duk da haka, kashi gyara an ba da ake bukata.

lokuta da yawan abin sama

Mene ne bayyanar cututtuka gani a marasa lafiya tare da "Oseltamivir" hakan allurai da miyagun ƙwayoyi? Reviews da kuma umarnin da cewa a ranar babu irin haka ya tashi. Duk da haka, guda dosages na antiviral magunguna zai iya sa amai ko kumallo.

Don warware wadannan cututtuka, symptomatic far.

Specific shawarwari domin samun magani

Me kana bukatar ka sani cikin haƙuri, kafin shan "Oseltamivir"? Umurnai na amfani (ga yara da kuma manya iya samun daban-daban illa) shi ya nuna cewa da miyagun ƙwayoyi ne ba m ga shekara-shekara alurar riga kafi. Ya bai hana ci gaban matsalolin da zasu iya faruwa a kwayar cututtuka, kazalika da kwayan cututtuka.

Analogs medicament

"Oseltamivir" - wani magani da cewa ne aka yi nufi ga jiyya da kuma rigakafin mura. Yana da wani antiviral wakili wadda ke da alaka hanawa na neuraminidase. Wannan magani an fiye da aka sani a karkashin iri sunan "Tamiflu". Tsarin analogs shi ba ya wanzu. A mafi kusa, amma dan kadan na baya yi, wadannan kwayoyi ne musanya, "Relenza", "Arbidol", "Flustol", "Kagocel" da sauransu.

Reviews da kimantawa da tasiri na da miyagun ƙwayoyi

Bisa ga gwajin sakamakon, wanda aka samu a Amurka da kuma Mexico, sabon ƙwayoyin cuta masu kula neuraminidase hanawa ( "Zanamivir" da "Oseltamivir"), amma su ne resistant zuwa wasu gungun - adamantanes ( "rimantadine", "Amantadine") .

Ya kamata kuma a lura da cewa masana da ba da inganci na wannan magani a lura da mura da aka shigar a cikin mutane tare da kullum zuciya da kuma numfashi cututtuka.

A cewar likitoci, da miyagun ƙwayoyi rage tsawon na cututtuka da 1 rana, amma wannan ne kawai da yanayin idan jiyya da aka fara a farkon 'yan sa'o'i bayan lamba tare da haƙuri.

Don kwanan wata, babu abin dogara bayani a kan ko tasiri na ci da miyagun ƙwayoyi a kan abin da ya faru na rikitarwa da kwayar ko cututtuka.

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