Kiwon lafiyaShirye-shirye

"Gabapentin" da kuma barasa: reviews. "Gabapentin": umarnin don amfani, haƙuri shedu da kuma likitoci

Daga lokaci zuwa lokaci, tsoka cramps dame mutane da yawa. Duk da haka, 'yan mutane tunani game da dalilin da ya sa irin wannan jihohin kullum tashi.

Bisa ga art, seizures iya zama daban-daban: jimlace (tonic, clonic, tonic-clonic da myoclonic) da kuma m (sauki da kuma hadadden). wani magani amfani da su bi seizures karshe a matsayin "Gabapentin". Umurnai na amfani, da sake dubawa kuma contraindications da miyagun ƙwayoyi za a gabatar kadan daga baya.

Ya kamata nan da nan a lura da cewa, ga m seizures halin da babu asarar sani. Irin wannan rare yanayin. Sun bayyana clonic seizures yanayi shafe wata tsoka hannayensu, feet da fuska.

Abun da ke ciki, description, marufi samfurin da kuma abun da ke ciki

sayar medicament "Gabapentin" A cikin me form? Shedu bayar da rahoton cewa wannan magani za a iya saya a kantin magani a cikin wani nau'i na tukuru gelatin capsules a fari. Da abun ciki shi ne wani farin ko yellowish foda miyagun ƙwayoyi.

The aiki sashi na wannan wakili ne gabapentin. Har ila yau, shi ya hada da wani ƙarin abu a cikin hanyar sodium carboxymethyl sitaci, alli stearate da microcrystalline cellulose. Amma ga capsules, suka dauke gelatin da titanium dioxide.

A wani kunshin sayar da miyagun ƙwayoyi "Gabapentin"? Mabukaci sake dubawa ce cewa a kan shelves na Pharmacy da miyagun ƙwayoyi za a iya samu a kwali fakitoci, wanda aka sanya ko dai polymeric capsules gwangwani ko kwane-kwane na cell.

A manufa na mataki na mai magani

Ta yaya miyagun ƙwayoyi "Gabapentin"? Umurnai (reviews na magani aka gabatar a karshen cikin labarin) rahoton cewa da miyagun ƙwayoyi a cikin tsarin ne sosai kama da neurotransmitter gamma-aminobutyric acid (Gaba for short). Duk da haka, ya kamata a lura da cewa manufa da ta mataki, ta sha bamban daga sauran kwayoyi da hulɗa tare Gaba-rabe (msl, valproate, barbiturates, benzodiazepines, Gaba transaminase hanawa, Gaba reuptake hanawa, Gaba agonists da prodrugs na Gaba).

An fito da miyagun ƙwayoyi yana da wani Gaba-ing Properties kuma ba zai tasiri a kama da metabolism na Gaba. Binciken masana sun nuna cewa aiki sashi daga cikin wakili da dauri ga α2-δ-subunit na ƙarfin lantarki dogara da alli tashoshi, ƙwarai rage da ya kwarara daga alli ions, wanda taka muhimmiyar rawa a farko na neuropathic zafi.

Features anticonvulsant miyagun ƙwayoyi

Abin da sauran kaddarorin ake mallaki by da miyagun ƙwayoyi "Gabapentin"? Reviews na likitoci sun ce yana da matukar tasiri ga neuropathic zafi. Wannan magani rage glutamate-dogara neuronal mutuwa, kara Gaba kira, kazalika da aiwatar da danniya na neurotransmitter saki da kuma monoamine kungiyoyin.

Ba za mu iya ce cewa a asibiti dacewa yawa daga miyagun ƙwayoyi "Gabapentin" ba daura wa rabe wasu kwayoyi (ko neurotransmitters), ciki har da Geba rabe da GABAB, kuma glutamate, benzodiazepine rabe, glycine, kuma N-methyl-D- aspartate.

Ba kamar "Carbamazepine" da "phenytoin", dauke da medicament ba hulɗa tare da sodium tashoshi. Shiri "gabapentin" partially attenuates sakamakon glutamate tsoka mai amsa sigina agonist kamar N-methyl-D-aspartate. Haka kuma, shi muhimmanci rage a saki monoamine neurotransmitters.

A sanadin motsi kaddarorin da miyagun ƙwayoyi

Mene ne muhimmi sanadin motsi sigogi capsules "Gabapentin"? Shedu ba za su iya amsa wannan tambaya. Don samun shi, za ku juya don gogaggen professionals ko a kewaye umarnin.

Bisa ga karshen, da bioavailability na ce kwayoyi ba su gwargwado ga sashi soma. Lokacin da adadin da miyagun ƙwayoyi ne rage.

A kan samun da medicament cikin iyakar jini taro lura bayan 3 h. A cikakkar bioavailability da miyagun ƙwayoyi a capsules ne kimanin 60%. Abinci, ciki har da mai ƙiba, yana da wani sakamako a kan motsi daga cikin miyagun ƙwayoyi.

Janyewar "Gabapentin" na haƙuri ta jini ne da za'ayi da wani mikakke model. rabin-rai lokaci ne mai zaman kanta da kashi kuma shi ne kamar 5-7 hours.

A sanadin motsi kaddarorin da miyagun ƙwayoyi ba ya canja ko da shi ne amfani da maimaitawa. A taro na miyagun ƙwayoyi a cikin jini za a iya annabta dogara ne a kan sakamakon da guda kashi.

A medicament "Gabapentin" ma ba ya daura wa jini sunadaran (kasa da 3%). An nuna a canzawa form ta kodan.

Metabolize da magani ake ba fallasa. Haka kuma, shi ba ya sa hanta oxidative enzymes, wanda suna da hannu a cikin metabolism na sauran kwayoyi.

The yarda da wakili daga jini rage-rage a mazan mutane da kuma marasa lafiya da sosai koda aiki.

Shiri "gabapentin" an cire daga jikin ta hemodialysis.

Alamomi sami magani

A abin da cututtuka muna la'akari da shi ne musamman tasiri magani? Abin da mutane suke cewa game da wannan feedback?

"Gabapentin" mai kyau bayyana kanta a cikin:

  • neuropathic zafi a adult marasa lafiya (18 shekaru da kuma mazan).
  • monotherapy ko matsayin karin magani domin lura da m seizures, tare da sakandare hakan a manya da matasa daga 12 shekara.

Contraindications don samun magani

Mene ne contraindications miyagun ƙwayoyi yana da "Gabapentin"? Reviews na aikace-aikace bayar da rahoton cewa yana da wani mummunan sakamako a jiki, idan magani an karɓa a:

  • hypersensitivity wa wani daga cikin abu.
  • m seizures karkashin yana da shekaru 12 years.

Special kula ne a wajen wajabta koda gazawar.

Ta yaya ya kamata in yi da magani "Gabapentin"?

Reviews (neuralgia wannan magani taimaka sosai kyau) jiha cewa da miyagun ƙwayoyi ya kamata a gudanar da kawai da wani gogaggen likita, bayan da daidai ganewar asali.

Gelatin capsules dauka baki ta hadiya dukan, a cikin form. A miyagun ƙwayoyi ya kamata a cinye ko na abinci, wanke saukar da m ruwa. Idan kana bukatar ka rage sashi na magani don soke ko maye gurbin ta analogue, to, wannan ya kamata a yi hankali, a hankali a mako.

Jiyya na neuropathic zafi a manya

Kamar yadda a wannan jiha ayyukan dauke magani? Abin da mutane suke cewa game da kiwon lafiya da sake dubawa? "Gabapentin" sosai yadda ya kamata bayyana kanta ga neuropathic zafi. A zalunta irin wannan yanayin na farko kullum kashi ya zama 900 MG. Ya ce adadin ne zuwa kashi uku rabo. Idan bukata, da kashi ne a hankali ya karu zuwa a kalla (Ina nufin, har zuwa 3600 MG da rana).

m seizures

Ta yaya ya kamata in yi da magani "gabapentin" a cikin wannan cuta? Reviews sun ruwaito cewa kayan aiki za a iya sanya ba kawai ga manya, amma matasa daga 12 shekaru.

A tasiri kashi ga m seizures dauke 900-2400 MG da rana. Jiyya da wannan cuta za su iya fara da 300 MG na da miyagun ƙwayoyi sau uku a rana. Daga bisani kullum kashi ya kamata a karu zuwa 900 MG, kuma mafi kuma har zuwa 2400 MG da rana (ya kasu kashi uku daidai allurai).

A lokaci tazara tsakanin allurai da miyagun ƙwayoyi a da sau uku liyafar kamata ba zama ya fi 12 hours (don kauce wa zaman majalisar na seizures).

illa

Abin da m halayen na iya faruwa a marasa lafiya samun anticonvulsant? Abin da mutane suke cewa game da wannan mabukaci reviews? "Gabapentin" da magani daga neuropathic zafi zai iya sa:

  • asthenia, mai haɗari rauni, da zafi na daban-daban sarrafawa, ciwon baya, kamuwa da cuta, mura ciwo, ciwon kai, nauyi riba, na gefe edema.
  • Gait tashin hankali, ataxia, ɓacin hankali, hypoesthesia, da ruɗewa, juwa ko jiri, illa tunani, drowsiness, tsãwa;
  • maƙarƙashiya, flatulence, zawo da amai, bushe baki, dyspepsia, tashin zuciya, ciwon mara.
  • fata rash.
  • shortness na numfashi, ciwon makogwaro.
  • amblyopia.

A lura da m seizures, da miyagun ƙwayoyi taimaka wa bayyanar:

  • ciwon baya, gajiya, zazzabi, ciwon kai, kwayar cutar, na gefe edema, nauyi riba, gajiya, malaise, fuska edema.
  • maƙarƙashiya, hakori cuta, zawo, bacin, ta ƙara ci, bushe baki ko makogwaro, tashin zuciya ko amai, ciwon mara, bloating, anorexia, gingivitis.
  • alama na vasodilation ko hauhawar jini.
  • leukopenia, purpura.
  • samu karaya, myalgia da arthralgia.
  • ɓacin hankali, ataxia, da ruɗewa, incoordination, ciki, dysarthria, wani tunanin lability, rashin barci, nervousness, nystagmus, drowsiness, mahaukaci tunani, tremor, tsoka twitching, juwa ko jiri, hyperkinesia. riba, weakening ko babu reflexes, juyayi, paresthesia, rashin jituwa.
  • abrasions, kuraje, fata itching, fata na gaggawa.
  • tari, pharyngitis, rhinitis, ciwon huhu.
  • amblyopia, diplopia, Heart hangen nesa.
  • urinary fili cututtuka, rashin ƙarfi.

lokuta da yawan abin sama

Mene ne bayyanar cututtuka na yawan abin sama na iya haifar da ce medicament? Me game da wannan ce da sake dubawa? "Gabapentin" yawan abin sama Yanã biyu hangen nesa, juwa ko jiri, drowsiness, illa magana, lethargy da zawo.

Don kawar da irin wannan jihohin symptomatic far, kazalika da aka azabtar wanke ciki da kuma ba shi kunna gawayi.

Marasa lafiya da tsanani na koda insufficiency, hemodialysis aka nuna.

Drug "Gabapentin" da barasa

Reviews kwararru bayar da rahoton cewa ya dace na dauke da kwayoyi ne sosai high. Amma shi ne kawai a cikin taron cewa lokaci na da aikace-aikace da haƙuri ne gaba daya watsi da amfani da giya.

Idan da miyagun ƙwayoyi ne a hade tare da barasa, da mãsu haƙuri iya muhimmanci worsen m halayen daga tsakiya m tsarin (mãyen, ataxia, da dai sauransu).

miyagun ƙwayoyi interactions

Drug "gabapentin" a neuroscience, reviews daga waxanda suke da fiye da kyau, za a iya hada ba tare da dukkan magunguna.

Bisa ga umarnin, antacids rage bioavailability da miyagun ƙwayoyi.

Myelotoxicity kwayoyi kara haematotoxicity capsules "Gabapentin".

Lokacin hade tare da morphine ta pharmacokinetics aka bai canja ba. Duk da haka, a lokacin da irin mai hade da ya kamata a hankali da sanya idanu m m dauki na juyayi tsarin.

An sano medicament iya dauka lokaci guda tare da antiepileptic kwayoyi (msl, "pentobarbital", "Carbamazepine", "Phenytoin" da kuma valproic acid) da kuma baka hana. A wannan yanayin, shi ba ya canja motsi.

takamaiman shawarwari

Duk da cewa da janyewar ciwo tare da ya faru na seizures da magani daga "gabapentin" da aka ba alama ta wani ba zato lõkacin fatara daga jiyya da antiepileptic kwayoyi a cikin mutane tare da m seizures iya har yanzu tsokane karfi convulsions.

An fito da magani ba wani tasiri wajen magance da rashi epilepsy.

Mutanen da suke bukatar hadaddun far da morphine, na iya bukatar wani ƙara kashi na "gabapentin". A wannan yanayin, tabbatar da m monitoring na haƙuri ga ci gaban drowsiness. A ta gano magunguna kashi ya kamata a mayalwaci rage.

Lokacin da hada "gabapentin" da sauran anticonvulsant kwayoyi da aka ruwaito ƙarya tabbatacce sakamakon a tabbatar da dalilin da furotin a fitsari amfani da gwajin tube Ames N-Multistix SG. A wannan batun, domin irin wannan nazarin bayar da shawarar yin amfani da wani takamaiman hazo Hanyar da sulfosalicylic acid.

Reviews kwararru da kuma masu amfani da

Mafi reviews na likitoci da marasa lafiya game da "Gabapentin" shiri ne tabbatacce. Wadannan rahotanni bayar da shawarar cewa da miyagun ƙwayoyi yadda ya kamata a magance da aiki. Duk da haka, idan aka hada tare da barasa sukan ci gaba mai tsanani m halayen a cikin juyayi tsarin.

Ba shi yiwuwa ba a lura da cewa ba zato karbo daga cikin miyagun ƙwayoyi iya haifar da marasa lafiya blunted sani, lethargy kuma mummunan yanayi.

Mutane da yawa sun lura da cewa, ci na wannan yana nufin suna da wata ciki da kuma bakin wake tunani. Har ila yau, magani sau da yawa yana sa da ci gaban m pancreatitis.

Masana sun bayar da shawarar zuwa miyagun ƙwayoyi jiyya "Gabapentin" kawai a karkashin kulawa na likita wanda zai iya sauri daidaita da warkewa regimen kamar yadda ake bukata.

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