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Da miyagun ƙwayoyi "Celebrex": reviews, analogs, umarnin don amfani, farashin

Da shan kashi na kashin baya, ciwo mai tsanani a cikin gidajen abinci da kuma connective nama canji ayyuka a kan bango na kumburi - rashin alheri, wadannan cututtuka sun fi na kowa a cikin lokaci. A wannan Jihar harkokin rinjayar salon, rashin al'ada jiki aiki, kwayoyin dalilai. Bugu da kari zuwa ciwo mai tsanani da cewa mutane wahala a wannan yanayin, rashin lafiya iya lalata dukan kwayoyin, musanyãwa jini sunadarai da shafi da al'ada aiki na kayan ciki.

Saboda haka muhimmanci wajen saka idanu da kiwon lafiya da kuma lokacin da za a yi wa cutar. Daya daga cikin mafi inganci da kwayoyi, wanda nasa ne da rukuni na ba-steroidal kwayoyi kira medicament "Celebrex". Reviews likitoci tabbatar da ingancinta a kwatanta da wannan layi na anti-kumburi kwayoyi.

Babban sakamako daga cikin miyagun ƙwayoyi

An yi amfani da miyagun ƙwayoyi iya kira da ikon hana kumburi tsari aiki a matakai daban-daban na cutar. Da zarar a cikin jini, da miyagun ƙwayoyi ne iya hana TSOG2 aiwatar da take kaiwa zuwa taimako na kumburi. "Celebrex" The miyagun ƙwayoyi yana da karfi analgesic dukiya antipyretic aiki. Saboda haka, yana ba kawai gusar da kumburi foci, amma kuma daidai kawar da ko da ciwo mai tsanani, rage zazzabi.

A abũbuwan amfãni daga wannan samfurin hada da kadan sakamako a kan platelets, cewa shi ne, da miyagun ƙwayoyi ba sa matsalolin da jini clotting. Lokacin da ka karɓi wani maras steroidal wakili cewa akwai wani hangula na ciki da kuma hanjinsu, rage hadarin ulcers da kuma gastritis marasa lafiya.

Saboda haka, "Celebrex" kwayoyi suna amfani da yawa more yadu fiye da sauran NSAID kwayoyi, "naproxen", "asfirin", "ibuprofen".

directional

"Celebrex" capsules suna da ikon rage tsananin hadin gwiwa zafi, stiffness kashe su jimre da matsanancin kumburi. Irin wannan daukan hotuna yiwu mu bi marasa lafiya bincikar lafiya tare da rheumatoid amosanin gabbai, osteoarthritis. Effect da miyagun ƙwayoyi kai matsakaicin sakamako ya 24-48 sa'o'i bayan da farko kashi. Dysmenorrhea miyagun ƙwayoyi yadda ya kamata gusar da zafi, ko da mafi m. Har ila yau, shi ne, yadda ya kamata amfani ga taimako na jin zafi bayan tiyata (maxillo-fuska da kuma orthopedic tiyata).

Marasa lafiya da ankylosing spondylitis miyagun ƙwayoyi "Celebrex" zai kawar da pathological tafiyar matakai da kuma inganta jiki ta ikon aiki. Lokacin da lura da muhimmancin iyalinmu adenomatous polyposis amfani da miyagun ƙwayoyi ya kai ga wani gagarumin raguwa a ci gaban da polyps a cikin ciwon da duodenum: rage adadin su kuma size. Doctors da'awar cewa isasshen allurai da magani da kuma riko da magani regimens iya cimma kyau kwarai da sakamakon da yin amfani da "Celebrex" miyagun ƙwayoyi. Shedu nuna kadan illa yayin da shan wannan magani.

A siffar da kuma abun da ke ciki na miyagun ƙwayoyi

Sosai zabe mai hanawa ne gelatin kwantena kusan fararen ko fari, ba su da m kuma alama da a blue tube suna "7767" a gefe daya da kuma "100" da "200" a kan sauran. Kwantena abinda ke ciki: granulated fari canza launi.

A abun da ke ciki na miyagun ƙwayoyi hada da: celecoxib (asali aiki sashi), lactose, povidone K30, sodium lauryl sulfate, magnesium stearate, sodium croscarmellose. A harsashi da aka yi da titanium dioxide, da kuma edible gelatin. Idan dace gwamnati da miyagun ƙwayoyi intramuscularly injections suna nada "Celebrex". Wannan irin magani aka sallami a cikin nau'i na bayani ga allura 2.2 ml ampoules - asali abu celecoxib.

Pharmacokinetics

Da miyagun ƙwayoyi da aka kyau tunawa a cikin jini a cikin azumi jihar, kuma ya kai a kalla yi bayan game da 2-3 hours. Duk da haka, da yin amfani da nufin tare da m abinci iya a jinkirta bayar da jari ga 1-2 hours. Saboda haka wajibi ne tuntubar likita game da lokacin shan magani.

Da zarar a cikin jini, da aiki abubuwa ba su ɗaure zuwa ja da maikacin jini, amma inji ba zai tasiri da nasara da ake so taro da miyagun ƙwayoyi a cikin jiki. Drug metabolized a cikin hanta da hadawan abu da iskar shaka da kuma glucuronidation shafe CYP2C9 enzyme. Fitarwa na nufin tare da fitsari da kuma tumbi a cikin nau'i na sauki metabolites, kuma kawai 3% na aiki abu ya zauna canzawa.

Drug "Celebrex", analogues daga waxanda suke da irin wannan a cikin abun da ke ciki, same wajen, haddasa kadan lalacewar kiwon lafiya, saboda iyawarsa da za a tunawa kamar yadda zai yiwu da kuma kusan gaba daya shafe ta daga jiki. Tare da wani low jiki nauyi lura da hakan taro na miyagun ƙwayoyi a cikin jini, kuma wannan sabon abu ne lura fiye a mata. Shi ba a san dalilin da ya sa, amma kuma a cikin mutanen da baƙar fata lura da wannan kuzarin kawo cikas. Saboda haka, wadannan kungiyoyi na marasa lafiya wajabta wani m kashi na magani a farkon far.

alamomi

Kamar yadda wani ba-steroidal anti-kumburi jamiái ga symptomatic magani wajabta miyagun ƙwayoyi "Celebrex". Alamomi ga yin amfani da:

  • rheumatoid amosanin gabbai.
  • osteoarthritis.
  • spondylitis.
  • algomenorrhea.
  • m zafi (post-dau lokaci, ciwon baya, musculoskeletal cututtuka).
  • amfani da magani daga adenamotoznogo polyposis.

Ya kamata a lura cewa isasshen magani iya kawai sanya wani likita a kan tushen da gudanar da bincike.

Hanyoyin da gwamnati da miyagun ƙwayoyi

Shan miyagun ƙwayoyi dole ne a ciki, ko da kuwa da abinci. Chewable Allunan kada ta kasance, kana bukatar ka sha bayyana ruwa. Ya kamata a lura da cewa zuciya da jijiyoyin jini rikitarwa iya faruwa da kullum gwamnati na da miyagun ƙwayoyi. Saboda haka, likitoci rubũta "Celebrex" a takaice hanya na lura. Guest masana tabbatar da cewa matsakaicin kashi ga dogon lokacin da magani ya kamata ba ƙetare 400 MG da rana!

  • Jiyya na osteoarthritis - isasshen kashi 200 ne MG da rana. Chance na guda kashi ko tsaga a cikin biyu (a yau da kullum jinkiri).
  • Rheumatoid amosanin gabbai - sa ran kashi na 100, ko 200 MG zuwa sau 2 a kowace rana. A lõkacin da mafi tsanani siffofin - har zuwa 400 MG sau biyu a rana.
  • Ankylosing spondylitis - 200 MG da rana, domin 1 ko 2 raba allurai. A likita ta hankali da kashi iya ƙara mayalwaci m
  • Dysmenorrhea da karfi zafi - ta fara far da 400 MG da rana da kuma kara da juna 200 MG a ranar farko na far, idan ya cancanta. A cikin wadannan kwanaki, dole ne ka dauki 200 MG sau biyu a rana.

Duration na lura ne m da halartar likita.

Contraindications da amfani da miyagun ƙwayoyi

Bugu da kari ya yiwu rashin lafiyan halayen ga yayan da miyagun ƙwayoyi, akwai hani a karkashin abin da aka haramta daga yin amfani da miyagun ƙwayoyi "Celebrex":

  1. Bronchial fuka, urticaria, rashin lafiyan da sauran NSAIDs.
  2. A postoperative lokaci bayan aortkoronarnogo kewaye.
  3. Peptic miki (exacerbation).
  4. GI zub da jini.
  5. Kumburi hanji cuta.
  6. Zuciya rashin cin nasara.
  7. Mai tsanani hanta insufficiency.
  8. Koda insufficiency.
  9. Pregnancy kuma lactation.
  10. Ba da shawarar don amfani a karkashin 18.
  11. Hypersensitivity ga yayan da miyagun ƙwayoyi da kuma sulfonamides.

Kariya kamata amfani da miyagun ƙwayoyi da ruwa riƙewa a cikin jiki, cututtuka na zuciya da jijiyoyin jini tsarin, da ciwon sukari.

illa

Duk da high iko da miyagun ƙwayoyi, da shafe tsawon ko ba daidai ba liyafar yanayin da sashi na iya zama illa da miyagun ƙwayoyi "Celebrex". Shedu nuna ya fi kowa (m) cututtuka kamar:

  • Rashin lafiyan halayen ciki har da kurji, urticaria, pruritus.
  • Flatulence, dyspepsia, edema, rashin barci.
  • Tari, rhinitis, mura-kamar dauki da kuma numfashi fili cututtuka.
  • Urinary fili cututtuka.

Da yawa kasa akwai ƙãra juyayi, anemia, tinnitus, flushes, arrhythmia, jijiya hauhawar jini. Wasu marasa lafiya da aka rubuta ulceration na narkewa kamar fili, angionevropatichesky edema, da samuwar bullae a kan fata, exacerbation na pancreatitis ko ta ci gaba, rikice. Duk wadannan cututtuka zai iya kawai faru ne lokacin da wani hanya na lura ne a takaicce (har zuwa 12 makonni, ba wucewa 800 MG da kashi). Amma a yanayin saukan dogon lokacin da magani (har zuwa shekaru 3) an lura:

  • Common: takaici da kujera, hauhawar jini, da ciwon ya kama daga cikin kunnuwa, angina, tsokar zuciya infarction, tashin zuciya, dysphagia, prostatitis, ta ƙara creatinine.
  • More rare: arrhythmia, angina, ischemic bugun jini, atherosclerosis, barci cuta, da bakin farji na jini, ulcers na bakin, dysmenorrhea, karuwa a haemoglobin, karu a hematocrit.

The hulda da miyagun ƙwayoyi da sauran kwayoyi

A medicament rayayye biotransformed shafe P450 2C9 (cytochrome). Saboda haka zai yiwu kai tsaye hulda da miyagun ƙwayoyi da sauran jamiái:

  1. Concomitant amfani da kwayoyi "Warfarin" na kara hadarin m zub da jini.
  2. Shiri "Ketanazol" da "Fluconazole" kara maida hankali na aiki abu celecoxib kusan ninki biyu.
  3. Karbar blockers ko ACE hanawa angiotenzita NSAIDs iya rage tasiri antigipertinzivny
  4. Hade kayayyakin dauke da lithium, shi zai iya muhimmanci ƙara da jini matakin.
  5. An haramta lokaci guda amfani da miyagun ƙwayoyi "Celebrex" analogs dauke da celecoxib, sauran NSAIDs!

miyagun ƙwayoyi analogues

Shi ne ya kamata a lura da cewa "Celebrex" miyagun ƙwayoyi halin kaka ba da yawa, da farashin ne a kan talakawan daga 400 zuwa 450 rubles. 10 capsules (100 MG sashi). Duk da haka, irin wannan magani ne quite tsada ga haƙuri da dadewa far. A wannan yanayin, da yarda daga likita, sanya jamiái dauke da celecoxib. Domin da miyagun ƙwayoyi "Celebrex" analogues na masu biyowa:

  • miyagun ƙwayoyi "Ranselak".
  • miyagun ƙwayoyi "Revmoksib".
  • Allunan "Flogoksib".
  • kwantena "Artoksib".

Wadannan analogs dauke da wannan aiki abu da kuma samun ma m warkewa sakamako da magani daga cututtuka. Ka lura da cewa wani isasshen kashi na wani analogue kuma sanya kawai da halartar likita. A wannan yanayin da likita ya wadãtu da daban-daban abun da ke ciki AIDS a analogs, suka dauke daban-daban Additives kamar yadda idan aka kwatanta da miyagun ƙwayoyi "Celebrex". Umarni sake bitar likitoci bayar da shawarar da yiwuwar wani rashin lafiyan dauki da mãsu haƙuri ga excipients na daban-daban magunguna daya kungiyar.

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