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"Paroxetine": umarnin don amfani, reviews. miyagun ƙwayoyi analogues

Abin da ake nufi da miyagun ƙwayoyi "Paroxetine"? Umurnai na yin amfani da miyagun ƙwayoyi za a gabatar a wannan labarin. Har ila yau daga gare shi, ka zama sane da kowane Contra-alamomi da suke samuwa daga wannan magani, idan ya na da wani sakamako masu illa, a cikin abin da nau'i ne samuwa da kuma yadda da miyagun ƙwayoyi interacts tare da wasu kwayoyi.

Abun da ke ciki, da kuma marufi nau'i na da miyagun ƙwayoyi saki

Drug "Paroxetine" ke sayarwa a cikin nau'i na alluna, film-mai rufi. Su madauwari kuma lenticular siffar, farin launi, da kuma hadarin wani m surface.

The aiki abu ne dauke da mu nufin paroxetine hydrochloride hemihydrate. Har ila yau, da miyagun ƙwayoyi a cikin abun da ke ciki yana da goyon bayan abubuwa a cikin nau'i na colloidal silicon dioxide, microcrystalline cellulose, crospovidone, alli hydrogen phosphate, copovidone, talc da magnesium stearate.

Allunan "Paroxetine" da aka sayar a bororo fakitoci na 10 guda wanda an sanya shi a cikin wani kwali akwatin.

A pharmacological mataki da miyagun ƙwayoyi

Mene ne magani "Paroxetine", wanda analogues za a mai suna dan kadan m? Yana da wani antidepressant. Yana da wani mai hanawa na (zabe) serotonin reuptake kwakwalwa neurons. Wannan shi ne abin da kayyade ta anti-depressive illa da kuma inganci da magani daga tsoro cuta da kuma m-na kullum cuta.

An duba lamba da medicament yana da matukar low dangantaka for α2-, α1- da β-adrenoreceptors kazalika da m-holinoretseptorami, dopamine, 5HT1-kamar, 5HT2-kamar kuma histamine H1-rabe.

Shin psychomotor ayyuka warware da miyagun ƙwayoyi "Paroxetine"? Reviews na likitoci sun ce da magani yana da wani sakamako a kan mutum psyche barnatar. Haka kuma, shi ba ya potentiate da depressant effects na ethanol a kan psychomotor ayyuka.

Wai masu bincike sun gano wani antidepressant irin wannan rauni Kunna Properties kawai idan an gudanar a dosages mafi girma fiye da wadanda ake bukata domin hanawa na serotonin reuptake. Ba za mu iya ce cewa wannan magani ba ya haifar da wani gagarumin canji a cikin jini matakan, EEG da kuma zuciya rate.

A pharmacokinetics wata na'urar kiwon lafiya da

miyagun ƙwayoyi "Paroxetine" kamar yadda tunawa? Umarnin don amfani, real likitoci sun ce bayan baka gwamnati na aiki abu da ake tunawa daga narkewa kamar fili da kuma aka metabolized ta cikin hanta.

A tsit taro na medicament a cikin jini samu ta hanyar 1-1.7 makonni bayan qaddamarwa na miyagun ƙwayoyi jiyya. The aiki sashi daga cikin miyagun ƙwayoyi ne a baje rarraba a kyallen takarda. A wannan yanayin, shi ne kawai kashi daya da aka samu a cikin jini. Sadarwa tare da sunadarai na domin na 95%.

Antidepressant metabolized a cikin hanta. A sakamakon haka, m metabolites suna kafa. Su sauri shafe ta daga jiki, da kuma samun low pharmacological aiki da kuma da wani sakamako a kan warkewa sakamakon da miyagun ƙwayoyi.

miyagun ƙwayoyi "Paroxetine" kamar yadda aka nuna? Lura, harhada magunguna ratings bayyana cewa game da 64% na aiki abu ne sallami tare da fitsari, yayin da sauran 36% - a cikin hanji (a bile).

A pharmacokinetics da miyagun ƙwayoyi a musamman na asibiti yanayi

A taro na aiki abu a cikin jini jini ƙaruwa a take hakkin da koda da hanta, kazalika da tsofaffi.

Alamomi ga yin amfani da wata na'urar kiwon lafiya da

A wasu lokuta, marasa lafiya suna wajabta antidepressant "Paroxetine"? a kan aikace-aikace na kayan aiki da jagora ya ƙunshi wadannan jerin karatu:

  • wani irin ciki, ciki har da mai tsanani na ciki, mai amsawa, kuma yana tare da tashin hankali.
  • tsoro cuta, ciki har da agoraphobia.
  • m-na kullum cuta (OCD ko rage tsawon).
  • kowa yana da tashin hankali cuta.
  • zaman juyayi rashin lafiya, ko ake kira social phobia.

Contraindications ga yin amfani da wata na'urar kiwon lafiya da

A wasu lokuta, a wani hali ba za a iya amfani da marasa lafiya antidepressant "Paroxetine"? a kan aikace-aikace na kayan aiki da jagora ya hada da wadannan jerin contraindications:

  • m epilepsy.
  • lokaci guda amfani da monoamine oxidase hanawa, kazalika da biyu-mako lokaci bayan janyewar.
  • yara shekaru.
  • gestation lokacin.
  • Hypersensitivity da miyagun ƙwayoyi aka gyara.
  • a lokacin shayarwa.

Yi amfani da matsananci hankali

A abin da lokuta kamata a sarrafawa ci daga antidepressant "Paroxetine"? Umurnai na amfani furta cewa, wannan shiri da aka gudanar tare da taka tsantsan don marasa lafiya da hanta gazawar, kwana-ƙulli glaucoma, koda gazawar, mania, benign prostatic hyperplasia, convulsive jihohi, cardiac cuta, epilepsy. Bugu da kari, cikin lokaci guda amfani da daidai ba magani da kuma cardioversion, kazalika da magunguna da cewa kara hadarin zub da jini. Ya kamata mu biya musamman da hankali ga gaban hadarin dalilai ga zub da jini cuta da kuma azama irin cuta jihohi.

Antidepressant "Paroxetine": da yadda za a sha maganin?

Muna la'akari da magani ake dauka baki daya a rana (da safe) a lokacin karin kumallo. Allunan ya kamata a yi lõma da dukan, wanke saukar da ruwa tare da bayyana.

A lokacin farko da makonni uku bayan da farkon magani da sashi ne gyara akayi daban-daban. An baya gyara (idan ya cancanta).

A lokacin shafe tsawon ciki da shawarar adadin da medicament ne 20 MG sau daya a rana. Idan bukata, da kashi ne a hankali ya karu da 10 MG. Max samu da miyagun ƙwayoyi kada wuce 50 MG.

Domin m na kullum cuta na farko kashi na wani antidepressant ne 20 MG da rana. Sa'an nan, yanã ƙara zuwa 10 MG. The shawarar talakawan kullum kashi ga wannan wata karkata ne 40 MG. A m larura shi za a iya ƙara zuwa 60 MG.

Idan haƙuri yana da wani tsoro cuta, za ka iya farko kai har zuwa 10 MG da miyagun ƙwayoyi a kowace rana. Don rage yiwu hadarin tsoro cututtuka a wani m kashi na da miyagun ƙwayoyi ne ya karu da 10 MG. A kan talakawan, a lokacin da irin wannan sabawa ne m don amfani 40 MG "paroxetine" a hours, matsakaicin yawan - 50 MG.

Lokacin da zamantakewa phobia ko zamantakewa tashin hankali cuta medicament farko ƙarfi kada wuce 20 MG da rana. Idan bayan irin wannan magani da ake so sakamako ba a cimma, sa'an nan makonni 2 da kashi ne a hankali ya karu zuwa matsakaicin, cewa ne har zuwa 50 MG da rana.

A jimlace tashin hankali cuta warkewa da kuma sa hannu girma daga cikin medicament ne 20 MG da rana

Idan haƙuri kamu da hanta ko koda gazawar, da shawarar kashi ya zama 20 MG da rana.

Mazan mutane a rana za a iya cinye babu fiye da 40 MG na magani.

Domin ya hana janyewar bayyanar cututtuka daina shan miyagun ƙwayoyi bada shawarar a hankali.

lokuta da yawan abin sama

Akwai lokuta da yawan abin sama da antidepressants kamar "Paroxetine", "Fluoxetine"? Masana sun lura cewa yin amfani da babban yawan kwayoyi suka gaske adversely shafi jikin mutum. A haƙuri kwarewa tashin zuciya, bushe baki, sinus tachycardia, amai, convulsions, tremor, bradycardia, mydriasis, agitation, irritability, sweating, nystagmus, ta ƙara jini, somnolence, kuma nodal kari.

A fairly rare lokutta yayin da yin amfani da miyagun ƙwayoyi da sauran psychotropic kwayoyi, da kuma barasa iya comatose haƙuri da bambancin da nuni a kan ECG. A tsanani yawan abin sama, da mãsu haƙuri ne serotonin ciwo da kuma rhabdomyolysis.

Abin da ya yi a irin wannan yanayi? A cikin hali na miyagun ƙwayoyi yawan abin sama "Paroxetine" ya zama na ciki da lavage, da kuma daukar kunna carbon. Idan dole, symptomatic magani.

illa

Mene ne illa na magani zai iya sa "Paroxetine"? Reviews na likitoci sun ce wannan kayan aiki da gaske taimaka wajen samar da wata matsala. Wadannan sun hada da wadannan yanayi da cututtuka:

  • A wani ɓangare na tsakiya m tsarin da kuma na gefe m tsarin: mania, drowsiness, da ruɗewa, tremor, serotonin ciwo, gajiya, hallucinations, rashin barci, nervousness, juwa ko jiri, depersonalization, gajiya, tsoro harin, seizures, agitation, ɓacin hankali, extrapyramidal cuta, myoclonus, tashin hankali.
  • Musculoskeletal tsarin: tsoka rauni, arthralgia, myopathy da myalgia.
  • Hankula: Heart da Heart hangen nesa a matsayin dukan.
  • Urinary tsarin: m urination ko urinary riƙewa.
  • Narkewa kamar fili: ƙãra ko rage ci, hepatitis, dandano canji, bushe baki, tashin zuciya, zawo da amai, da kuma maƙarƙashiya.
  • Haihuwa tsarin: anorgasmia, jima'i tabarbarewa, hyperprolactinemia ko galactorrhea, rashin ƙarfi da kawowa cuta.
  • Zuciya da jijiyoyin jini tsarin: orthostatic hypotension.
  • Alerji: itching, rash, angioedema, kuma urticaria, ecchymosis.
  • Sauran bambancin: rhinitis, sweating, bai dace ba mugunya antidiuretic hormone, hyponatremia.

Hulda da sauran likita nufin

A lokaci daya amfani da antacids ba zai tasiri a pharmacokinetic sigogi da sha da miyagun ƙwayoyi "Paroxetine".

Contraindicated ga daya-lokaci amfani da kudi kafin mu tare da Mao hanawa.

Lokaci daya liyafar medicament "paroxetine" tare da kwayoyi da hana hanta enzymes, na bukatar da ragewan na farko kashi.

Antidepressant tsawanta zub da jini a kan bango na daya-lokaci amfani "na warfarin."

Lokaci daya amfani da medicament "paroxetine" tare da tricyclic antidepressants, asfirin, atypical neuroleptics, NSAIDs kuma yana nufin phenothiazine jerin inganta jini clotting tsari.

Lokaci daya gwamnati da serotonergic jamiái (kamar "tramadol" da "sumatriptan") iya kai wa ga inganta serotonergic effects.

Yana da muhimmanci a tuna da!

Don kauce wa ci gaban da wani neuroleptic ciwo (m), wani magani da matsananci taka tsantsan "Paroxetine" wajabta wa marasa lafiya da suke suna shan antipsychotics.

Mazan mutane a kan bango da miyagun ƙwayoyi iya ci gaba hyponatremia.

Lokacin da na farko ãyõyin seizures da kuma mania antidepressant far aka tsaya.

A lokacin farko makonni na lura da "paroxetine" na bukatar da hankali da lura da na haƙuri saboda yiwu kashe kansa.

A lokacin far kamata shan giya saboda su inganta mai guba sakamako.

Katafaren amfani

Drug "Paroxetine" ba a wajabta wa yara, kamar yadda da aminci da kuma inganci a lura da marasa lafiya a cikin wannan kungiyar ba, an kafa.

Antidepressant "Paroxetine": takwarorinsu

Da miyagun ƙwayoyi za a iya maye gurbinsu "Paroxetine"? Ya kamata a lura cewa wannan magani, akwai quite 'yan takwarorinsu. Daga gare su, zai zama kyawawa mu haskaka da wadannan kwayoyi: "Reksetin", "Adepress", "Pliz", "Apo-Paroxetine", "Aktaparoksetin", "Paxil", "sertraline", paroxetine hydrochloride hemihydrate, "" Sirestill "da sauransu.

Don saya duk da wadannan magunguna a cikin kantin magani, ba za ka iya kawai ta sayen magani.

Reviews na medicament

Drug "Paroxetine" yana mai yawa gauraye da sake dubawa, duka daga kwararru da kuma daga marasa lafiya. A daya hannun, shi ne yabe su da abin da shi na taimaka wa m kawar da duk wani nau'in ciki (ciki har da mai tsanani na ciki, mai amsawa, kuma yana tare da tashin hankali), kazalika da tsoro, m-na kullum, kowa yana da kuma zamantakewa-tashin hankali cuta. A kan wasu - da yawa marasa lafiya ce cewa nan da nan bayan da miyagun ƙwayoyi da suka ci gaba quite babban yawan m halayen. A sakamakon haka, mutane sun ma yana da dakatar da magani.

A general, masana lura cewa "Paroxetine" - wannan shi ne mai matukar tasiri da ingantaccen magani copes tare da aiki sanya shi. Duk da haka, shi za a iya amfani ne kawai ga manufar da aka nufa gwani.

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