Kiwon lafiyaShirye-shirye

"Monosan": umarnin don amfani, real takwarorinsu

Me kuma a cikin abin da sashi wajabta da miyagun ƙwayoyi "Monosan"? Umurnai na yin amfani da vasodilator kwayoyi da aka bayyana a cikin daki-daki, a cikin kayan da wannan labarin. Har ila yau, shi ya gabatar da medicament analogs, abun da ke ciki, pharmacological effects, contraindications, illa, da sauransu. D.

A siffar, marufi, abun da ke ciki

Abin da abubuwa bangare ne na miyagun ƙwayoyi "Monosan"? Umarni ya furta cewa, yanzu kashi na wannan miyagun ƙwayoyi ne isosorbide-5-mononitrate. Har ila yau, medicament qunshi wani abun da ke ciki da kuma irin adjuvants: talc granulated lactose, magnesium stearate, microcrystalline cellulose da masara sitaci.

A abin da fom masana'antun sarrafa miyagun ƙwayoyi "Monosan"? Umurnai na amfani jihohin da wani magani za a iya sayi kawai a cikin nau'i na alluna. Su ne fari da kuma zagaye a siffar. A gefe daya daga cikin kwamfutar hannu akwai hadarin.

Da miyagun ƙwayoyi ne kunsasshen a blisters, wanda aka located a cikin tari na kwali.

pharmacological siffofin

Ta yaya miyagun ƙwayoyi "Monosan"? Umurnai na amfani na nuni da cewa da miyagun ƙwayoyi ne a gefe vasodilator, wanda abubuwa da farko a kan venous tasoshin.

A medicament ne iya ta da samar da jijiyoyin bugun gini endothelium endothelial shakatawa factor kamar nitrogen oxide. A sakamakon irin wannan effects ne kunnawa da narkewa guanylate cyclase (kwayuka enzyme) cewa ta kanta qara vasodilating matsakanci - cyclic guanosine monophosphate.

Bayan shan miyagun ƙwayoyi a ciki Kwayoyin rage tsokar oxygen bukatar. Wannan shi ne saboda wani karu a yi da kuma post-preload.

Har ila yau, kwararru sun rajista a pronounced sakamako koronarorasshiryayuschee magani.

miyagun ƙwayoyi effects

Abin da sauran miyagun ƙwayoyi yana da kaddarorin "Monosan"? A amfani da wannan magani zai iya rage jini ya kwarara da dama atrium, wanda muhimmanci rage matsa lamba a cikin huhu wurare dabam dabam da kuma rage tsanani daga cikin mummunan cututtuka na huhu edema.

Ya kamata kuma a lura da cewa, a karkashin tasirin "Monosana" a yankunan da matalauta zagayawa akwai wani redistribution na jijiyoyin zuciya jini ya kwarara

A kan bango da miyagun ƙwayoyi a cikin mutane tare da angina kuma ischemic cututtukan zuciya, muhimmanci ƙara juriya da duk wani jiki aiki. Bugu da kari, batun wakili ne iya rage da CA sigogi Thrombocyte kira da kuma hana platelet tari.

pharmacokinetic Properties

Inda shi ne tunawa, rarraba da metabolized miyagun ƙwayoyi "Monosan"? Umarnin a kan aikace-aikace jihohi da cewa mataki na miyagun ƙwayoyi abu wajen sauri da kuma cikakken tunawa daga narkewa kamar fili. Bayan samun Allunan antianginal sakamako da aka lura bayan kamar minti 30-45 da kuma kiyaye domin 10 hours.

A cewar kwararru, da miyagun ƙwayoyi "Monosan" yana da wani fairly high kudi na bioavailability (kamar 99-100%). Wannan shi ne saboda babu farko izinin da miyagun ƙwayoyi ta hanyar da hanta tsarin.

A rabin rai da miyagun ƙwayoyi ne 60 minutes. A taro na miyagun ƙwayoyi a cikin jini dabam dan kadan, dangane da mutum.

Metabolism da kwayoyi aiki dũkiyõyinsu a cikin hanta. A sakamakon tafiyar matakai na rayuwa suna kafa na uku aka gyara: isosorbide glucuronide da biyu isosorbide-5-mononitrate.

rabin-rai lokaci ne 4-5 hours. Lokacin da wannan 2.2% da aka excreted via da na koda tsarin da 97,8% - kamar yadda glucuronic metabolites.

alamomi

A karkashin abin da yanayi da ake sa wa "Monosan"? A amfani da wannan magani ne mafi tasiri a cikin wadannan lokuta:

  • na huhu hauhawar jini, na huhu zuciya.
  • kullum siffofin congestive zuciya rashin cin nasara.
  • stenokardicheskie rigakafin seizures a mutane da jijiyoyin zuciya jijiya cuta.

contraindications

A karkashin abin da yanayi ba za a iya amfani da "Monosan"? Analogs kuma ce yana nufin kanta an haramta da za a dauka a lokacin da:

  • jijiyoyin bugun gini auka.
  • a Jihar buga.
  • jijiya hypovolemia da hypotension.
  • cardiac tamponade .
  • bar na ramin zuciya kasawa da kuma low fihirisa na diastolic jini;
  • mai guba na huhu edema.
  • m lokaci na tsokar zuciya infarction (tare da pronounced hypotension).
  • fom-ƙulli glaucoma.
  • nono.
  • cututtuka da cewa tsokana Yunƙurin na intracranial matsa lamba;
  • mutum hypersensitivity.
  • a cikin yara da matasa (har zuwa shekaru masu rinjaye).

Ya kamata kuma a lura da cewa, rahoto na nufin akwai zumunta contraindications. Wadannan yanayin ya shafi su:

  • mitral stenosis .
  • constrictive pericarditis.
  • tsufa.
  • jijiyoyin bugun gini cuta orthostatic tsari.
  • koda insufficiency tsarin.
  • hypertrophic cardiomyopathy.
  • hyperthyroidism.
  • hanta gazawar ;
  • aortic stenosis.
  • m anemia cikin.

Drug "Monosan": umarnin don amfani da

INN (International Nonproprietary Name) da wannan magani sauti kamar "isosorbide mononitrate." Wannan magani an gudanar da baki kawai. Bisa ga umarnin, ya kamata a yi lõma da dukan da kuma wanke saukar da ruwa.

Allunan kamata sanya wani likita. A lokaci guda ya zamar masa dole domin tantance mai tsanani daga cikin tamkar cuta da ya haƙuri.

"Monosanom" Jiyya farawa da karža yana nufin 10-20 MG 1-3 a rana sau. Tare da 3-4 kwanaki na far sabawa ya kamata a yi dosing regimen. Idan dole, yawan miyagun kwayoyi ya karu zuwa 20-40 MG da kuma shan sau biyu a kowace rana.

bayyanar cututtuka na yawan abin sama

Mene ne alamun yawan abin sama na iya faruwa a lokacin da wani haƙuri samun da ba daidai ba magani "Monosan"? Umurnai na amfani nuna da wadannan cututtuka: auka, aka rufe da mãgãgi, zawo ciwo, juwa ko jiri, hyperpnoea, redness na fata, da jarirai, dyspnea, tachycardia reflex asalin, ciwon kai, pyrexia, lethargy, wani rauni, ta ƙara intracranial matsa lamba, na gani disturbances, seizures, inna, tashin zuciya, coma, sweating, amai.

A zalunta irin wannan yanayi kamar yadda aka yi amfani da sabawa ciki lavage kuma rubũta enterosorbiruyuschee nufi.

illa

Shin m miyagun ƙwayoyi dauki "Monosan"? Umurnai na amfani (analogs na medicament aka nuna a kasa) ya tanadi cewa irin wannan magani na iya haifar da bayyanar da wani jam'i na gefe-effects. Mun ambaci wasu daga cikinsu:

  • amai.
  • kona abin mamaki a kan harshen.
  • bushe baki.
  • tashin zuciya.
  • zafi filasha.
  • tachycardia.
  • nitrate ciwon kai.
  • yankin Flushing da fata .
  • dizziness.
  • alama raguwa a jini.
  • stenokardicheskie ya karu mita na seizures.
  • Orthostatic hypotension .
  • hypersomnia.
  • shafi tunanin mutum retardation da kuma mota martani.
  • stiffness.
  • Heart hangen nesa.
  • kafa haƙuri.
  • takamaiman fata rashes.
  • exfoliative dermatitis.

Analogs na miyagun ƙwayoyi da ta price

Wanda ke nufin ba za ka iya canza magani «Monosan"? Analogues na wannan magani da ake samu a kowane kantin magunguna. Daga cikin mafi tasiri ne mai yiwuwa a ware "Monocinque gudanar", "Izoket", "Kardiket", "Efoksa", "Pektrol".

Kamar yadda ga farashin da miyagun ƙwayoyi, shi ne ba sosai high. Saya miyagun ƙwayoyi a Rasha birane iya kawai ga 100s (30 Allunan).

shedu

muna la'akari da miyagun ƙwayoyi yana mai yawa tabbatacce feedback. Marasa lafiya jayayya da cewa behaves kamar yadda mai matukar tasiri wakili don na huhu hauhawar jini da kuma na kullum zuciya maye siffar. Duk da haka, ya kamata a lura da cewa domin samun high warkewa sakamakon irin wannan magani ya kamata a hade tare da sauran kwayoyi. Don yin wannan, a tabbatar tuntubar da halartar likita.

Ina kuma so a lura da cewa da yawa marasa lafiya so farashin ƙaddamar da miyagun ƙwayoyi. Kamar yadda aka ambata a sama, 30 Allunan za ka biya kawai 100 Rasha rubles.

Ba za mu iya ce cewa game da miyagun ƙwayoyi da kuma sau da yawa bar mummunan feedback. A mafi yawan lokuta, su suna hade da bayyanar da wani jam'i na gefe-effects. Af, a lokacin da suka faru daga ingestion ya kamata a yi watsi da kuma maye gurbinsu da more amintacce wajen. Me daidai, za ka iya gaya kawai wani gogaggen gwani.

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