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Da miyagun ƙwayoyi "Papaverin". Bayanin zai taimaka wajen amfani da su

Daga cikin kwayoyi da dama da aka amince da su a cikin shekaru masu yawa a marasa lafiya, akwai magani kamar "Papaverin." Umarnin ya bayyana dalla-dalla duk alamun da maganin amfani da wannan alkaloid. A cikin yanayi, wannan abu yana dauke da opium. Kwanan nan, an samar da shi a lokaci-lokaci. Wannan abu abu ne mai nauyin katako, mai sauƙi a cikin barasa, mai narkewa cikin ruwa. Foda yana da ɗanɗɗo mai ɗanɗano. Maganin ruwa mai mahimmanci na abu shine haifuwa na tsawon awa 0.5 a zafin jiki na 100 ° C.

Drug "papaverine" yana nufin miotropnym antispasmodic. Ya rage aiki na kwangila kuma ya rage sautin miki tsokoki, yana da aikin antispasmodic da vasodilating. Wannan shiri da ake amfani da matsayin antispasmodic a lokacin da mai santsi tsoka spasm (ga cholecystitis, pilorospazme, spastic colitis, spasms na urinary fili), na gefe jijiyoyin bugun gini, Bronchial, kwakwalwa tasoshin. Har zuwa kwanan nan, ana amfani da wannan magani don hana hare-haren angina pectoris. Samun maganin "Papaverin", abin da aka koya game da abubuwan da ke da nasaba da kyau, ya kamata a tuna cewa a cikin babban allurai yana hana ƙin intracardiac, ya rage karfin zuciyar tsoka. Miyagun ƙwayoyi suna rage karfin jini.

Kodayake likitocin sun rubuta magunguna "Papaverin" ga marasa lafiya, koyarwar ba ta ce ba a fahimci ma'anar aikinsa a jikin mutum ba. Wannan abu ne mai hanawa na phosphodiesterase, wani enzyme wanda ke haifar da kwayar halitta tara na cyclic adenosine monophosphate. Ƙungiyarta tana haifar da raguwa a cikin kwangila na musculature da kuma shakatawa a lokacin yanayi na spastic.

Sau da yawa, tare da tare da promedolom sanya wani magani "Papaverin", wanda ake ba da izinin yin amfani da shi tare da wasu kwayoyin antispasmodic da analgesic. Irin wannan farfadowa an yi don kawar da hare-haren angina pectoris. Har ila yau an rubuta wannan magani a hade tare da platyphylline, phenobarbital da sauran abubuwa.

An saki miyagun ƙwayoyi "Papaverin" a cikin Allunan (0.04 g) a cikin kunshe na kwakwalwa 10., A cikin ampoules tare da bayani na 1 da 2% na 2 ml, a cikin kwakwalwan zane na 0.2 g. Abin da ke aiki a cikin Allunan, sauƙin shiga cikin tarihin Ganyayyaki, da sauri shiga cikin ƙwayar narkewa. Ana amfani da miyagun ƙwayoyi ta kodan. Rabin rabin rayuwa daga rabin sa'a zuwa 2 hours. Har zuwa kashi 60 cikin dari na maganin wannan abu an sake shi ta hanyar nau'in mahaukaci (tare da glucuronic acid, phenolic).

Magungunan miyagun kwayoyi "Papaverin", wanda ya bayyana a fili abin da allurai zai dauki magungunan miyagun ƙwayoyi ga marasa lafiya na shekaru daban-daban, yana buƙatar kulawa da waɗannan ka'idoji. Jimalar wucewa yakan haifar da mummunan sakamako. Manya a kowace rana yawanci an umarce su sau 3-4 a magani na 1 kwamfutar hannu (0.04 g). Sanya kwayoyi ga yara, dangane da yawan shekarun, don yin amfani da lokaci 3-4 a cikin irin waɗannan abubuwa:

- 0,5-2 shekaru: 0,25-0,5 Allunan;

- 3-4: 0.5-1 tebur;

- 5-6: 1 tebur;

- 7-9: 1.5 Allunan;

- 10-14: 1,5-2 shafin.

Intramuscularly da kuma karkashin fata bayani allura zuwa 1-2 ml (1; 2%). Hankali da kuma sannu a hankali gudanar a cikin jijiya 2% bayani (2.1 ml), kamar yadda da miyagun ƙwayoyi zai iya sa da ya faru na atrioventricular block, na ramin zuciya fibrillation da kuma na ramin zuciya extrasystoles. A cikin nau'i na kwarewa, wakili yana amfani da 0.003-0.03 g da kashi (sashi yana dogara da shekaru). Ana amfani da kyandirori bayan yin amfani da kwasfa ko kuma motsi.

Shan magani contraindicated da hypersensitivity cikinta, hypotension, take hakkin atrioventricular madugu. Kada ka dauki miyagun ƙwayoyi ba tare da tuntubi likita ba. Ƙarfafawa ko kiyaye lafiyar shi a lokacin lactation da ciki ba a kafa. Sabili da haka, maganin "Papaverin", alamun da ake amfani dashi a wannan lokacin bai zama mahimmanci ba, yana da kyau kada yayi amfani da shi. A lokacin magani, ba a yarda da barasa ba.

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