Kiwon lafiyaShirye-shirye

Da miyagun ƙwayoyi "Akineton": umarnin don amfani, description, reviews

The aiki abu "Akinetona" ne biperiden hydrochloride. Tablet ruwansa 2 MG na aiki abu. Bugu da ƙari, kasancewar ƙarin aka gyara (masara sitaci, dankalin turawa, sitaci, lactose monohydrate, magnesium stearate, microcrystalline cellulose, copovidone, alli hydrogen phosphate dihydrate, talc, da ruwa mai tsarkakẽwa) kwakwalwa gaba da miyagun ƙwayoyi "Akineton".

Umurnai na amfani, da photo nuna cewa kwamfutar hannu tsari da miyagun ƙwayoyi yana da kusan farin launi, Valium form. A gefe daya daga cikin kwamfutar hannu akwai hadarin wani beveled giciye siffar.

1 ml na bayani ƙunshi biperiden lactate a wani adadin na 5 milligrams. Ƙarin aka gyara su ne: alura ruwa da kuma sodium lactate.

pharmacological effects

Babban sashi biperiden - holinoblokator tsakiyar mataki.

A tasiri shafi yanã raunanar da ikon cholinergic neuronal aiki a cikin striatum, wanda shi ne tsarin naúrar na extrapyramidal tsarin.

Da miyagun ƙwayoyi sa ganglioblokiruyuschimi sakamako, antispasmodic kuma matsakaici mai tsanani m-anticholinergic effects a periphery (antispasmodic).

Amfani da miyagun ƙwayoyi taimaka kashe reshe tremor, wanda ya taso a cikin yin amfani da cholinergic kwayoyi (msl, pilocarpine) da kuma catalepsy da tsoka rigidity a marasa lafiya samun neuroleptics. Yana da ikon sa agitation.

Pharmacokinetics

"Akineton" daure su jini da sunadarai a 91-94%. Jini yarda zai zama 11.6 ± 0.8 ml / min / kg jiki nauyi. A guda kashi na baka halitta yana mai bioavailability na game da 33 ± 5%.

Wuce a cikin nono.

Biperiden cikakken metabolized a cikin jikin mutum. A fitsari, da abu ba m, a sãkẽwa form. Manyan metabolites ne bicycloheptane da piperidine, wanda suke fitarwa daga tumbi da fitsari.

Elliminatsiya za'ayi a biyu bulan, da rabin rayuwa (T 1/2) na minti 90 a lokacin da farko lokaci da kuma 24 hours - na biyu lokaci. A tsofaffi da marasa lafiya, da rabin-rai za su iya kara ma.

alamomi

"Akineton" amfani da extrapyramidal cuta jawo by gwamnati na wasu magunguna (neuroleptics, antipsychotics).

Har ila yau, da miyagun ƙwayoyi ne nuna ga ganewar asali na cutar Parkinson ta ciwo, parkinsonism (wakili gudanar a hade far da wani tushe)

contraindications

Manufar wannan miyagun ƙwayoyi ba a nuna a lokacin da kake hypersensitive da aiki sashi daga cikin miyagun ƙwayoyi "Akineton".

Umurnai na amfani sanar da cewa da miyagun ƙwayoyi kamata a kauce masa a cikin ganewar asali da cuta a cikin wani haƙuri kamar prostate kara girma, kwana-ƙulli glaucoma, obstructive canje-canje a cikin hanji (pylorus stenosis, shanyayyen ileus Farawa).

Arrhythmia, epilepsy, nono ciyar, tsofaffi, ciki ne dalilai a wadda "Akineton" gudanar da a yi taka tsantsan.

illa

CNS illa an bayyana asthenia, gajiya, lethargy, wani rauni, numbness, juwa ko jiri, ji na damuwa, tashin hankali, memory hanawa, da ruɗewa, hallucinations, catalepsy, miyagun ƙwayoyi dogara miyagun ƙwayoyi "Akineton".

Umurnai na amfani magana game da gefen-illa da kuma tare da wani ɓangare na hangen - mydriasis, tashin hankali na masauki.

Cardio-jijiyoyin bugun gini tsarin ne halin da quickening na zuciya rate (tachycardia). wani lokacin - deceleration (bradycardia). lokacin da ake ji allura nau'i na cikin shirye-shiryen - rage-rage a jini (hypotension).

A kan wani ɓangare na narkewa kamar tsarin - bushe baki, dyspeptic cututtuka, maƙarƙashiya.

A kan wani ɓangare na metabolism - rage sweating.

A wani ɓangare na urinary tsarin - a marasa lafiya tare da kara girma (hypertrophy) na prostate gland shine yake - yiwu wahala yana yin fitsari.

Rashin lafiyan halayen: kurji a kan fata, itching.

Hanyoyin da Amfani

Domin intramuscular, igiyar jini, da kuma da baka kwamfutar hannu tsari ne fit shiri "Akineton".

Umarnin don amfani da shawara cewa far "Akinetonom" kullum yana farawa daga kananan allurai, da kashi fiye da stepwise ƙaruwa dangane da ake so warkewa sakamako da kuma ga illa.

Manya a yin amfani da wata baka nau'i na shirye-shiryen fara jiyya a kashi na 1 MG 1-2 liyafar lokacin da rana ko 2 MG kasu kashi biyu allurai da rana. Bugu da ari, da sashi za a iya ƙara zuwa 8 MG biyu zuwa hudu raba allurai. Duk da haka, kashi kamata ƙãru ba, fiye da 2 MG da rana. Kada ku ƙẽtare iyakar sashi na nufin 6 cikin Th-16 MG kwanaki biyar. Single kashi injectable miyagun ƙwayoyi form kada wuce 2.5-5 MG. Wannan kashi iya maimaita bayan rabin sa'a, amma da yawan gwamnatocin da rana kada wuce sau 4. A kalla kashi na medicament a injectable nau'i ne 20 MG kwanaki biyar. Lokacin da mafi kyau duka kashi da aka kai, sa'an nan a miƙa mulki ga liyafar "Akinetona retard."

Amma kar ka manta game da mutum tsarin kula da kowane haƙuri a cikin saduwa biperidenom far.

Extrapyramidal Pathology tasowa saboda ingestion na wasu magunguna (antipsychotics ko neuroleptics) na bukatar aiki na wani ba abu a guda kashi na 2 MG baki ko parenterally. Maimaita gwamnati na ce allurai iya zama kowane awa daya da rabi. Duk da haka, kamar yadda aka nuna a bisa, da yawan gwamnatocin kada wuce sau 4. The baka kashi kamata a raba daya zuwa uku allurai.

Parkinson ta cuta shafi gudanarwa ta da miyagun ƙwayoyi da baki a 6-8 MG a 2-4 raba allurai domin a rana, da kashi za a iya hankali ya karu har zuwa 6-16 MG.

Yara a karkashin shekara nufi da shawara da yiwuwar daga cikin miyagun ƙwayoyi a cikin injectable form sannu a hankali, guda kashi na 1 MG ko 0.2 ml. Lokacin da shekaru daga shekara guda zuwa shekara shida gudanar 2 MG ko 0.4 ml. Daga 6 zuwa shekaru 10 - 3 MG ko 0.6 ml. Wannan kashi iya maimaita bayan rabin sa'a tare da gaggawa. A gaban illa a kan gwamnati da miyagun ƙwayoyi ya zama katse allura.
A lokacin da na baka nau'i na da miyagun ƙwayoyi far a shekaru daga 3 zuwa 15 shekaru na shan da sashi na 1-2 MG a 1-3 hours lokacin da rana.

Allunan ba zai iya sha a kan komai a ciki, kuma dole ne ka sha matsakaiciya yawan ruwa. A abin da ya faru na ke so illa daga narkewa kamar tsarin tafii da miyagun ƙwayoyi nan da nan bayan da wani abinci, rage tsanani daga cikin m tasiri nufin "Akineton".

Umurnai na amfani na nuni da cewa a cikin hali na nicotine guba a manya misali hadaddun far an kuma gudanar da wannan miyagun ƙwayoyi, da kuma ta kashi ne 5-Th-tarin fuka-10 MG ga injectable siffofin, amma kawai a lokuta da cewa barazana da haƙuri ta rayuwa.

Lokacin da guba kwayoyin phosphorus garwayayye biperiden dosing ne da za'ayi akayi daban-daban dangane da tsananin daga raunuka. Fara daga wani kashi na 5 MG a cikin hali na igiyar jini gwamnati, maimaita gwamnati ci gaba har sai da cututtuka bace guba.

yawan abin sama

Yawan abin sama bayyana pronounced anticholinergic effects sa da magani "Akineton".

Umarnin don amfani, real likitoci biya da hankali ga gaskiyar cewa maganin wannan yanayin posimptomnaya (gyaran zuciya da jijiyoyin jini da kuma na numfashi tsarin, oxygen far, hyperthermia gyara, a urinary catheter sa, idan ya cancanta). Bukatar gabatarwar a cholinesterase hanawa (physostigmine farko) .

hulda

"Akineton" yayin da amfani da m-holinoblokatorami, kwayoyi da ciwon wani antihistamine da antiepileptic mataki kara habaka magana na karshen. Duk da haka, lokaci daya aikace-aikace na metoclopramide rage da warkewa sakamako. Akwai tabbatacce miyagun ƙwayoyi incompatibility da ethanol. Ganawa quinidine ƙaruwa a sau da hadarin tasowa dyskinesia bayyanar cututtuka. M-cholinergic sakamako ne inganta lokacin da ake ji levodopa.

Storage da sayarwa

Don saya wannan magani na bukatar takardar sayen magani don samar da harhaɗa magunguna. Don adana "Akinetona" bukatar cika da zazzabi, t. E. yanayi zazzabi kada wuce 25 digiri (Celsius sikelin). Muna bukatar da isar yara da makaman "Akineton".

Manual bada shiryayye rai da miyagun ƙwayoyi - shekaru biyar.

tsõratar

Nada biperiden a lokacin daukar ciki da kuma nono (lactation) na bukatar m alamomi.

Biperiden iya samun zuwa jariri ta hanyar nono, haifar da wani wucin gadi gazawar da nono ga an daina miyagun ƙwayoyi "Akineton".

Samfurin description nuna cewa a yankan shawara a kan nada biperiden a lokacin daukar ciki da kuma lactation la'akari da hadarin m zuwa jariri, tayi.

Tsofaffi zama wani hadarin factor domin lura da wannan magani. Saboda haka sanya "Akineton" wannan rukuni na mutane da a yi taka tsantsan.

Kickaha babu wata shaida da yin amfani da jami'an tsaro a cikin shimfiɗar jariri, shi ne dalilin da cewa ba ya shafi miyagun ƙwayoyi yara "Akineton".

Description of shiri (umurci manual) ƙayyade da cewa hankali ake bukata a lokacin da yin amfani da wannan magani a marasa lafiya tare da epilepsy ko fibrillation.

Tare da shafe tsawon amfani iya ci gaba da miyagun ƙwayoyi dogara.

A hadarin karbo ciwo unshi da hankali lõkacin fatara daga far "Akinetonom".

da yin amfani da barasa-dauke da abubuwan sha kamata a kauce masa a lokacin far.

Jiyya tare da wannan magani na bukatar abstinence daga tuki motocin da wasanni ayyukan da bukatar babban taro da kuma m psychomotor halayen, tun da shi daukawa da shi da yuwuwar hadari saboda hadarin juwa.

"Akineton". Umarnin don amfani. analogs

Kamancin shiri ne da wadannan abubuwa: "Biperiden" "Mendileks" "biperiden hydrochloride".

"Akineton". reviews

A miyagun ƙwayoyi ne sosai tasiri a lura da Parkinsonism tremors a reshe da aka kare bayan wani gajeren lokaci tazara. Ya ce da kyau-jure magani "Akineton".

Feedback a kan forums magana game da yiwuwar bayyanuwar wasu illa yayin da shan miyagun ƙwayoyi.

Price "Akinetona". inda saya

A kudin da mafita iya zama a kusa da 800 rubles.

Price baka halitta "Akinetona" - 560-580 rubles.

Similar articles

 

 

 

 

Trending Now

 

 

 

 

Newest

Copyright © 2018 ha.delachieve.com. Theme powered by WordPress.