Kiwon lafiyaShirye-shirye

Naiz (kwamfutar hannu) - umurci manual.

sashi fom

A shirye-shiryen da aka sanya a cikin 3-miyagun ƙwayoyi siffofin - dakatar, dispersible Allunan, kuma na al'ada. The dakatar ne mai dadi wari tare da ambato rawaya a launi da kuma quite halayyar dandano na wannan magani. A dakatar da za a iya redispersed ta girgiza vial.

Allunan kerarre kusan fararen, tare da kadan yellowish tinge. Allunan na madauwari siffar, biconcave, ta biyu saman ne santsi.

Nise abun da ke ciki:

dakatar

Active abu

  • Nimesulide - 50 MG (5 ml na dakatar)

Excipients:

  • sorbitol
  • glucose
  • xanthan danko
  • propyl
  • methylparaben
  • citric acid
  • abarba dandano
  • Yellow fenti WS
  • glycerol
  • polysorbate
  • tsarkake ruwa

dispersible Allunan

Active abu

  • Nimesulide - 50 MG (Table 1).

excipients

  • aspartame
  • alli phosphate
  • microcrystalline cellulose
  • carboxymethyl sitaci
  • masara sitaci
  • talc
  • magnesium stearate
  • Colloidal silicon dioxide
  • abarba dandano

Allunan

Active abu

  • Nimesulide - 100 MG (Table 1).

Excipients:

  • magnesium stearate
  • Alli hydrogen Phosphate
  • microcrystalline cellulose
  • Anhydrous colloidal silicon
  • masara sitaci
  • Sodium sitaci glycolate
  • tsarkakakku talc

A pharmacological mataki da miyagun ƙwayoyi

Pharmacological mataki da dangantaka da farko zuwa Nise - kwayoyi, da wa'azi ƙunshi data for duk sashi siffofin. Da miyagun ƙwayoyi ne a NSAID, dauke da cikin da tsarin sulfonilidnuyu ra'ayoyi. Nimesulide Mayu da dangantaka da hanawa na Cox-2, sabõda haka, shi yana da anti-mai kumburi da analgesic effects, a Bugu da kari, da miyagun ƙwayoyi exerts analgesic effects, amma zuwa karami mataki.

Ginshikai na mataki na miyagun ƙwayoyi hade da danniya na kira na prostaglandins a kumburi da kuma danniya da samuwar oxygen radicals da kuma hanawa na myeloperoxidase saki.

Pharmacokinetics

Nise daidai tunawa daga cikin gastrointestinal fili, kai ta matsakaicin a cikin jini riga bayan 2 hours. A miyagun ƙwayoyi ne 99% gina jiki a ɗaure.

Shiri nize - Allunan jagora wanda aka dauka daga hukuma kafofin, metabiliziruetsya a cikin hanta da kuma excreted a cikin fitsari, tare da 98% na kashi samu ne fitarwa a lokacin da rana.

shaidar

  • Rheumatic cututtuka da cewa ci gaba wajen hadin gwiwa kwantena
  • osteoarthritis
  • Kumburi da kuma zafi bayan tiyata
  • Pain lalacewa ta hanyar dysmenorrhea
  • Fever da kuma zafi a lokacin m kumburi a cikin sama Airways

Side effects Nise

Allunan, da wa'azi ga wanda yanzu shi ne, za a iya samar da gefen-effects a daban-daban da kuma tsarin gabobin:

Side effects da miyagun ƙwayoyi, wanda dangantaka da narkewa kamar fili

  • tashin zuciya
  • ƙwannafi
  • ciki zafi
  • dakata stools

Side effects da miyagun ƙwayoyi, wanda dangantaka da tsakiya m tsarin:

  • ciwon kai
  • drowsiness
  • dizziness

Side effects da miyagun ƙwayoyi, wanda lãbãri a gare rashin lafiyan halayen:

  • erythema
  • rash
  • urticaria

Sauran gefen effects:

  • Riƙewa a cikin jiki ruwa
  • oliguria
  • ƙaruwa

Nise contraindications

An jerin contraindications a wadda ta bada shawarar don kauce wa shan miyagun ƙwayoyi, da kuma lokacin da cikakken zama dole, kawai bayan tuntubar likita.

  • Zub da jini daga gastrointestinal fili
  • koda gazawar
  • hanta gazawar
  • Pregnancy kuma lactation
  • Peptic gastrointestinal cuta

Drug hulda nize

Allunan, umarnin a kan yin amfani da abin da ba ya haifar da cikakken kuma m bayanai a kan dukkan miyagun ƙwayoyi interactions halitta ne kamar haka: ba da shawarar da wadannan jamiái - phenytoin, digoxin, wani diuretics, kwayoyi lithium, anticoagulants, antihypertensive kwayoyi, NSAIDs, methotrexate, cyclosporin .

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